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Validated Methods
Bioanalytical Laboratory Validated Bioanalytical Methods

July 2009
(*Latest methods and changes are highlighted.)

Drug LOQ, ng/mL Technique Matrix
Acetaminophen 100 LC-MS Human Plasma
Acyclovir 20 HPLC-FL Human Plasma
Amitriptyline 1 HPLC-UV Human Plasma
Amitriptyline 0.4 LC-MS/MS Human Plasma
Nortriptyline 0.4    
Amlodipine 0.1 LC-MS/MS Human Plasma
Anastrozole 0.1 LC-MS/MS Human Plasma
Atenolol 12.8 HPLC-FL Human Whole Blood
Atomoxetine 2.001 LC-MS/MS Human Plasma
4-Hydroxyatomoxetine 1.937    
N-Desmethylatomoxetine 1.999    
Atorvastatin 0.4 LC-MS/MS Human Plasma
o-hydroxyatorvastatin 0.4    
p-hydroxyatorvastatin 0.04    
Azithromycin 5 LC-MS Human Plasma
Betamethasone 0.5 LC-MS/MS Human Plasma
Betamethasone Acetate/ 0.5    
Betamethasone Phosphate 2    
Bromazepam 5 HPLC-UV Human Plasma
Bumetanide 1 HPLC-FL Human Plasma
Bupropion 1.0 LC-MS/MS Human Plasma & Rat Plasma
Bupropion Erythroamino Alcohol 1.0    
Bupropion Threoamino Alcohol 1.0    
Hydroxybupropion 4.0    
Bupropion 5.0 LC-MS/MS Rat Plasma
Bupropion Erythroamino Alcohol 1.0    
Bupropion Threoamino Alcohol 1.0    
Hydroxybupropion 2.0    
Buprenorphine 0.1 LC-MS/MS Human Plasma & Dog Plasma
Norbuprenorphine 0.1    
Buspirone 0.05 LC-MS/MS Human Plasma & Mouse Plasma
1-(2-Pyrimidyl)Piperazine 0.2    
Buspirone 0.4 LC-MS/MS Human Plasma & Rat Plasma
1-(2-Pyrimidyl)Piperazine 1.6    
Buspirone 0.039 LC-MS/MS Human Plasma
1-(2-Pyrimidyl)Piperazine 0.156    
6-Hydroxybupropion 0.625    
Carbamazepine 50 HPLC-UV Human Plasma
Carbamazepine-10, 11-Epoxide 10    
Carvedilol 1 LC-MS/MS Human Plasma
O-Desmethylcarvedilol 0.2    
4'-Hydroxyphenylcarvedilol 0.2    
5'-Hydroxyphenylcarvedilol 0.2    
Cefaclor 200 HPLC-UV Human Plasma
Cefixime 100 HPLC-UV Human Plasma
Cefuroxime 200 HPLC-UV Human Plasma
Celecoxib 20 HPLC-FL Human Plasma
Cephalexin 200 HPLC-UV Human Plasma
Chlorpheniramine 0.1 LC-MS/MS Human Plasma
Chloropheneramine 0.1 LC-MS/MS Human Plasma
Citalopram Chiral (R and S) 0.25 LC-MS/MS Human Plasma
Demethylcitalopram (R and S) 0.2    
Didemethylcitalopram (S) 0.2    
Cilazapril 1 LC-MS/MS Human Plasma
Cilazaprilat 0.250    
Cilazapril 4 LC-MS/MS Human Plasma
Cilazaprilat 1.000    
Ciprofloxacin 24.999 HPLC-FL Human Plasma
Ciprofloxacin 1500 HPLC-UV Human Urine
Desethyleneciprofloxacin 500    
Sulfociprofloxacin 500    
Oxociprofloxacin 500    
Formylciprofloxacin 500    
Cimetidine 12.5 HPLC-UV Human Plasma
Citalopram 0.25 HPLC-FL Human Plasma
Citalopram 0.25 LC-MS/MS Human Plasma
Demethylcitalopram 0.05    
Didemethylcitalopram 0.05    
Citalopram 0.25 LC-MS/MS Human Plasma
Demethylcitalopram 0.126    
Didemethylcitalopram 0.025    
Clarithromycin 20 LC-MS Human Plasma
Clavulanic Acid 100 LC-MS/MS Human Plasma
Clonazepam 0.1 LC-MS/MS Human Plasma
Clonidine 0.03 LC-MS/MS Human Plasma
Cloxacillin 100 HPLC-UV Human Plasma
Clozapine 0.1 LC-MS/MS Human Plasma
Cyproterone Acetate 0.3 LC-MS/MS Human Plasma
Ethinyl Estradiol 0.015    
Dextromethorphan/ 0.1 LC-MS/MS Human Plasma
Dextrorphan/ 1    
Pseudoephedrine 1    
Didanosine 10 LC-MS/MS Human Plasma
Diflunisal 500 HPLC-UV Human Plasma
Diltiazem 3 HPLC-UV Human Plasma
Desacetyldiltiazem 1    
N-Desmethyldiltiazem 3    
Diltiazem 0.781 LC-MS/MS Human Plasma
Desacetyldiltiazem 0.195    
N-Desmethyldiltiazem 0.391    
Diphenhydramine 0.5 LC-MS/MS Human Plasma
Doxazosin (achiral) 0.5 HPLC-FL Human Plasma
Doxepin 2 HPLC-UV Human Plasma
Nordoxepin 1    
Doxycycline 80 HPLC-UV Human Plasma
Duloxetine 0.5 LC-MS/MS Human Plasma
Dutasteride 40 LC-MS/MS Human Plasma
Efavirenz 0.02 LC-MS Human Plasma
Enalapril 0.25 LC-MS/MS Human Plasma
Enalaprilat 0.25    
Eprosartan 5 LC-MS/MS Human Plasma
Etodolac 250 HPLC-UV Human Plasma
Exemestane 0.2 LC-MS/MS Human Plasma
Exemestane 0.05 LC-MS/MS Human Plasma
Famotidine 5 HPLC-UV Human Plasma
Felodipine 0.05 LC-MS/MS Human Plasma
Fenofibric acid 10 HPLC-UV Human Plasma
Fenofibric acid 49.996 HPLC-UV Human Plasma
Fentanyl 0.02 LC-MS/MS Human Plasma
Fexofenadine 5 HPLC-FL Human Plasma
Fluconazole 100 HPLC-UV Human Plasma
Fluoxetine 0.5 LC-MS Human Plasma
Norfluoxetine 0.5    
Flupenthixol 0.1 LC-MS/MS Human Plasma
Fluticasone Propionate 0.001 LC-MS/MS Human Plasma
Fluticasone Propionate 0.005 LC-MS/MS Human Plasma
Fluvastatin 1.999 LC-MS/MS Human Plasma
Fluvoxamine 0.5 LC-MS/MS Human Plasma
Gabapentin 74.988 LC-MS/MS Human Plasma
Galantamine 0.5 LC-MS/MS Human Plasma
Ganciclovir 30 HPLC-FL Human Plasma
Gatifloxacin 25 HPLC-FL Human Plasma
Glimepiride 2 LC-MS/MS Human Plasma
Glipizide 2.5 LC-MS/MS Human Plasma
Glyburide 2 LC-MS Human Plasma
Griseofulvin 15 LC-MS/MS Human Plasma
Granisetron 0.02 LC-MS/MS Human Plasma
Guaifenesin 10 LC-MS Human Plasma
Hydrochlorothiazide 5 LC-MS Human Plasma
Hydrocodone 0.4 LC-MS/MS Human Plasma
Hydrocodone+Ibuprofen 1.0/100 LC-MS/MS Human Plasma
Hydromorphone 1    
Hydromorphone 0.05 LC-MS/MS Human Plasma
Ibuprofen 400 HPLC-UV Human Plasma
Indapamide 12.6 HPLC-UV Human Plasma
Indapamide 10 HPLC-UV Human Whole Blood
Indomethacin 10 HPLC-UV Human Plasma
Itraconazole 2.0 LC-MS/MS Human Plasma
Hydroxy Itraconazole 2.0    
Ketoprofen 300 HPLC-UV Human Plasma
Lamotrigine 20 HPLC-UV Human Plasma
Lansoprazole 2 LC-MS/MS Human Plasma
Leuprolide 0.025 LC-MS/MS Human Plasma
Letrozole 0.5 LC-MS/MS Human Plasma
Levetiracetam 0.5 LC-MS/MS Human Plasma
Lisinopril 0.25 LC-MS/MS Human Plasma
Lisinopril 1 LC-MS/MS Human Plasma
Loperamide 0.05 LC-MS/MS Human Plasma
Loratadine 0.1 LC-MS/MS Human Plasma
Descarboethoxyloratadine 0.1    
Loratadine/Pseudoephedrine 0.1/2.5 LC-MS/MS Human Plasma
Descarboethoxyloratadine 0.1    
Losartan 4.010 LC-MS/MS Human Plasma
Losartan Hydroxy Acid 3.998    
Lovastatin 0.1 LC-MS/MS Human Plasma
Lovastatin Hydroxy Acid 0.1    
Medroxyprogesterone Acetate 0.02 LC-MS/MS Human Plasma
Mefenamic acid 50 HPLC-UV Human Plasma
Megestrol Acetate 1 LC-MS/MS Human Plasma & Dog Plasma
Meloxicam 30.0 HPLC-UV Human Plasma & Dog Plasma
Meloxicam 1 LC-MS/MS Human Urine
Metaxalone 5 LC-MS Human Plasma
Metoprolol 1 LC-MS/MS Human Plasma
Metformin 10 LC-MS/MS Human Plasma
Metformin 2 LC-MS Human Urine
Methylprednisolone 0.4 LC-MS/MS Human Plasma
Metoprolol 2.5 HPLC-UV Human Plasma
Mirtazapine 0.5 LC-MS/MS Human Plasma
Misoprostol Acid / Diclofenac 0.01/19.997 LC-MS/MS Human Plasma
Mycophenolate Mofetil 0.04 LC-MS/MS Human Plasma
Mycophenolic Acid 100    
Nabumetone metabolite (6-MNA) 500 HPLC-FL Human Plasma
Nadolol 0.5 HPLC-FL Human Plasma
Nadolol/Bendroflumethiazide 2.000/1.000 LC-MS/MS Human Plasma
Naltrexone 0.1 LC-MS/MS Human & Dog Plasma
6-ß-Naltrexol 0.1    
Naltrexone 1.0 LC-MS/MS Human Urine
6-ß-Naltrexol 10    
Naproxen 500 HPLC-FL Human Plasma
Nefazodone 6.25 LC-MS Human Plasma
2-Hydroxynefazodone 1.88    
m-Chlorophenylpiperazine 1.25    
Nifedipine 0.5 LC-MS/MS Human Plasma
Nifedipine 0.5 LC-MS or LC-MS/MS Human Plasma
Nitrofurantoin 20 HPLC-UV Human Plasma
Nizatidine 10 HPLC-UV Human Plasma
N-Desmethylnizatidine 5    
Nortriptyline 1 HPLC-UV Human Plasma
Norfloxacin 20 HPLC-FL Human Plasma
Omeprazole 1 LC-MS/MS Human Plasma
Ondansetron 0.5 LC-MS/MS Human Plasma
Oxaprozin 1000 HPLC-UV Human Plasma
Oxcarbazepine 10 LC-MS/MS Human Plasma
10,11-dihydro-10-Hydroxycarbamazepine 50    
Oxycodone 0.5 LC-MS/MS Human Plasma
Noroxycodone 0.5    
Oxymorphone 0.1    
Oxybutynin 0.16 LC-MS/MS Human Plasma
Desethyloxybutynin 1.56    
Oxymorphone 0.04 LC-MS/MS Human Plasma
Hydroxy Oxymorphone      
Pantoprazole 20.001 LC-MS Human Plasma
Paroxetine 0.2 HPLC-FL Human Plasma
Paroxetine 1.563 HPLC-FL Human Plasma
Pentoxifylline 1.3 LC-MS/MS Human Plasma
Hydroxy Pentoxifylline 4.3    
and CPDX 4.3    
Phenylephrine (Total) 4 LC-MS/MS Human Plasma
Phenytoin 40 HPLC-UV Human Plasma
Pindolol 2 HPLC-FL Human Plasma
Pramipexole 0.04998 LC-MS/MS Human Plasma
Pravastatin 0.25 LC-MS/MS Human Plasma
3-a-Hydroxy Pravastatin 0.25    
Pravastatin 1 LC-MS/MS Human Plasma
3-a-Hydroxy Pravastatin 1    
Prazosin 0.1 HPLC-FL Human Plasma
Primidone 200 LC-MS/MS Human Plasma
Phenobarbital 200    
Phenylethylmalonamide 200    
Propranolol 0.4 HPLC-FL Human Plasma
4 -Hydroxypropranolol 0.8    
Quetiapine 1 LC-MSMS Human Plasma
Ramipril 0.05 LC-MS/MS Human Plasma
Ramiprilat 0.05    
Ranitidine 25 HPLC-UV Human Plasma
Risedronate 0.2 LC-MS/MS Human Plasma
Rosiglitazone 1.996 LC-MS/MS Human Plasma
Sertraline 0.25 LC-MS/MS Human Plasma
N-Desmethylsertraline 0.25    
Simvastatin 0.1 LC-MS/MS Human Plasma
Simvastatin Hydroxy Acid 0.1    
Sotalol 10 HPLC-FL Human Plasma
Sirolimus 0.4 LCMSMS Human Plasma
Sulfamethoxazole 200 HPLC-UV Human Plasma
Trimethoprim 20    
Sulfasalazine 20 LC-MS Human Plasma
Sulfapyridine 200    
5-Aminosalicylic acid 20    
Acetyl-5-aminosalicylic acid 10    
Sumatriptan 0.5 LC-MS/MS Human Plasma & Pig Plasma
Tacrolimus 0.2 LC-MS/MS Human Whole Blood
Tamoxifen 0.25 LC-MS Human Plasma
n-Desmethyltamoxifen 0.25    
Tamoxifen 0.25 LC-MSMS Human Plasma
Tamsulosin 0.05 LC-MS/MS Human Plasma
Terazosin 0.5 HPLC-FL Human Plasma
Terbinafine 10 HPLC-UV Human Plasma
Theophylline 150 HPLC-UV Human Plasma
Ticlopidine 10 HPLC-UV Human Plasma
Topiramate 5 LC-MS/MS Human Plasma & Dog Plasma
Topiramate 50 LC-MS/MS Human Plasma
Torsemide 10.0 LC-MS/MS Human Plasma
Tramadol 2.0 LC-MS/MS Human Plasma & Mouse Plasma
O-Desmethyltramadol 1.0    
O,N-di-Desmethyltramadol 1.0    
Tramadol 195 LC-MS/MS Human Urine
O-Desmethyltramadol 49    
O,N-di-Desmethyltramadol 49    
Tramadol 2.0 LC-MS/MS Human Plasma & Dog Plasma
O-Desmethyltramadol 1.0    
Tramadol 2.001 LC-MS/MS Human Plasma
Meloxicam 3.750    
O-Desmethyltramadol 1.000    
O,N-di-Desmethyltramadol 1.000    
Trazodone 10 HPLC-FL Human Plasma
Triamcinolone acetonide 0.5 LC-MS/MS Human Plasma
Trimebutine 0.999 LC-MS/MS Human Plasma
N-Desmethyltrimbutine 9.981    
Valproic acid 924 HPLC-UV Human Plasma
Valsartan 20 LC-MS/MS Human Plasma
Venlafaxine 1 LC-MS/MS Human Plasma
O-Desmethylvenlafaxine 2    
N-Desmethylvenlafaxine 1    
N,O-Didesmethylvenlafaxine 1    
N,N,O-Tridesmethylvenlafaxine 1    
Venlafaxine 100 LC-MS/MS Human Urine
O-Desmethylvenlafaxine 200    
N-Desmethylvenlafaxine 100    
N,O-Didesmethylvenlafaxine 200    
N,N,O-Tridesmethylvenlafaxine 101    
Verapamil (Chiral ) 1.6 HPLC-FL Human Plasma
Norverapamil R and S 1.6    
Verapamil 2 HPLC-FL Human Plasma
Norverapamil 2    
Vigabatrin 0.2 LC-MS Human Plasma
Warfarin (R-Warfarin) 1 LC-MS/MS Human Plasma
S-Warfarin 1    
Ziprasidone 0.125 LC-MS/MS Human Plasma
Zolpidem 1 HPLC-FL Human Plasma

 

 

 

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